Scalarane-based sesterterpenoid RCE-protease inhibitors isolated from the Indonesian marine sponge Carteriospongia foliascens.

نویسندگان

  • David E Williams
  • Irwin Hollander
  • Larry Feldberg
  • Eileen Frommer
  • Robert Mallon
  • Akbar Tahir
  • Rob van Soest
  • Raymond J Andersen
چکیده

Two new 20,24-bishomo-25-norscalaranes, compounds 1 and 2, and two new and two known 20,24-bishomoscalaranes, compounds 3-6, have been isolated from the Indonesian marine sponge Carteriospongia foliascens. The structures of 1-6 were determined by spectroscopic analysis. Compounds 1 and 3-6 inhibit RCE-protease activity.

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Cytotoxic scalarane sesterterpenoids from the South China Sea sponge Carteriospongia foliascens.

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عنوان ژورنال:
  • Journal of natural products

دوره 72 6  شماره 

صفحات  -

تاریخ انتشار 2009